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12 NEW KINASE INHIBITORS RELEASED |
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| Bafetinib |
| SYN-1179 |859212-16-1 |
| Bafetinib (INNO-406) is a potent and selective dual Bcr-Abl, Lyn inhibitor with IC50 of 5.8 nM and 1... |
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| NVP-BGT226 |
| SYN-1178 |1245537-68-1 |
| NVP-BGT226 is a novel, orally bioavailable small-molecule inhibitor of phosphoinositol-3-kinase and ... |
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| (+)-JQ1 |
| SYN-3004 |1268524-70-4 |
| (+)-JQ1 is a potent, high affinity, selective BET bromodomain inhibitor (IC50 values are 17.7, 32.6,... |
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| Vorinostat |
| SYN-3006 |149647-78-9 |
| Vorinostat inhibits the activities of HDAC1 and HDAC3 with IC50 of 10 nM and 20 nM, respectively.... |
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| GNF-5837 |
| SYN-1183 |1033769-28-6 |
| GNF-5837 is a potent, selective and orally bioavailable pan-TRK inhibitor of TRKA, TRKB and TRKC wit... |
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| CX6258 |
| SYN-1182 |1202916-90-2 |
| CX6258 was reported to be the potent inhibitors of Pim-1, Pim-2 and Pim-3 kinase inhibitor with IC50... |
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| Latest News |
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Synkinase Newsletter Jan 2013_VEGFR
It was reported that AVEO Oncology and Astellas Pharma have begun enrolling patients with advanced t... |
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NEW Warehouse in US. Providing next day Delivery
Synkinase has opened a warehouse in San Diego California.
We will provide next day delivery.
Call ... |
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SynKinase Newsletter: December 12 2012
A kinase interaction map profiling the activity of 178 commercially available kinase inhibitors agai... |
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SynKinase Newsletter in November 2012: Kinase Inhibitor Selectivity
Protein kinases represent the most important classes of therapeutic targets because of their pivotal... |
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